Durroux, T.

Time-Resolved FRET Binding Assay to Investigate Hetero-Oligomer Binding Properties: Proof of Concept with Dopamine D1/D3 Heterodimer

G protein-coupled receptors (GPCRs) have been described to form hetero-oligomers.

Hounsou, C.

• Feb 20, 2015 • 1 min read

Selective Fluorescent Nonpeptidic Antagonists For Vasopressin V2 GPCR: Application To Ligand Screening and Oligomerization Assays.

A series of fluorescent benzazepine ligands for the arginine–vasopressin V2 receptor (AVP V2R) was synthesized using “Click” chemistry.

Loison, S.

• Oct 25, 2012 • 1 min read

Mapping the Binding Site of Arginine Vasopressin to V1a and V1b Vasopressin Receptors

Starting from the 2.

Rodrigo, J.

• Feb 1, 2007 • 1 min read

Key Amino Acids Located within the Transmembrane Domains 5 and 7 Account for the Pharmacological Specificity of the Human V1b Vasopressin Receptor

In mammals, the vasopressin V(1b) receptor (V(1b)-R) is known to regulate ACTH secretion and, more recently, stress and anxiety.

Derick, S.

• Nov 1, 2004 • 1 min read